7.下列抗生素中,何者抗菌機轉不是抑制細菌之蛋白質合成,以達到bacteriostatic或bactericidal effects?
(A)quinupristin-dalfopristin
(B)tedizolid
(C)tigecycline
(D)fosfomycin
答案:登入後查看
統計: A(1228), B(532), C(413), D(3809), E(0) #3135874
統計: A(1228), B(532), C(413), D(3809), E(0) #3135874
詳解 (共 10 筆)
#5905038
來自阿摩前人的整理:
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#6036747

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#6149389
pristin結尾抑制蛋白合成
cycline 結尾為四環類抑制蛋白合成(抑制ribosome)
olid結尾也是抑制蛋白質合成
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抑制核酸多為xacin, azole, ximin(x常出現)結尾
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這題還算沒有陷阱,出現兩個mycin或者故意出Lincomycin, Clindamycin就刺激了
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比較需要特別注意mycin結尾
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1. Cell Wall Synthesis Inhibitors (細胞壁合成抑制劑)
- Beta-lactams (β-內醯胺類):
- Penicillins (青黴素類): Amoxicillin, Ampicillin, Penicillin G
- Cephalosporins (頭孢菌素類): Ceftriaxone, Cefazolin, Cephalexin
- Carbapenems (碳青黴烯類): Imipenem, Meropenem
- Monobactams (單醯胺環類): Aztreonam
- Glycopeptides (糖肽類):
- Vancomycin (萬古黴素)
- Teicoplanin
- Lipoglycopeptides:
- Telavancin
- Dalbavancin
- Oritavancin
- Fosfomycin (磷黴素):
- Fosfomycin
2. Protein Synthesis Inhibitors (蛋白質合成抑制劑)
- Aminoglycosides (胺基糖苷類):
- Gentamicin (慶大黴素)
- Tobramycin (妥布黴素)
- Amikacin (阿米卡星)
- Tetracyclines (四環素類):
- Tetracycline (四環素)
- Doxycycline (多西環素)
- Minocycline
- Tigecycline
- Macrolides (巨環內酯類):
- Erythromycin (紅黴素)
- Azithromycin (阿奇黴素)
- Clarithromycin (克拉黴素)
- Lincosamides:
- Clindamycin
- Oxazolidinones (噁唑烷酮類):
- Linezolid (利奈唑胺)
- Tedizolid
- Streptogramins:
- Quinupristin/dalfopristin
- Chloramphenicol (氯黴素):
- Chloramphenicol
3. Nucleic Acid Synthesis Inhibitors (核酸合成抑制劑)
- Quinolones (喹諾酮類):
- Ciprofloxacin (環丙沙星)
- Levofloxacin (左氧氟沙星)
- Moxifloxacin (莫西沙星)
- Rifamycins (利福黴素類):
- Rifampin (利福平)
- Rifabutin
4. Cell Membrane Disruptors (細胞膜破壞劑)
- Polymyxins (多黏菌素類):
- Polymyxin B (多黏菌素B)
- Colistin
- Lipopeptides:
- Daptomycin
5. Folic Acid Synthesis Inhibitors (葉酸合成抑制劑)
- Sulfonamides (磺胺類):
- Sulfamethoxazole (磺胺甲噁唑)
- Trimethoprim (甲氧苄啶):
- Trimethoprim
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